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  • 原料藥及中間體服務

    吉林天衡原料藥和中間體生產基地位于河南省鄧州市工業園區南陽天衡制藥廠,車間占地1萬平米,各類型反應釜40余臺。依托北京天衡藥物研究院有限公司產品的研發 ,已完成小試品種有100多個,目前工業化規模生產13個品種,產品質量達到國際高水平。產品出口日本、印度、東南亞和歐洲部分國家。


    原料藥及中間體服務產品目錄



    產品名稱Product nameCAS登記號(CAS No.)標準Specification結構式Structural Formula
    伏格列波糖及中間體
    Voglibose & Intermediates
    伏格列波糖
    Voglibose
    83480-29-9JP16
    IP
    In house
     01
    2,3,4,6-四-O-芐基-α-D-葡萄糖
    2,3,4,6-Tetra-O-benzyl-α-D-glucopyranose
    4132-28-9
    6564-72-3
    ≥99%
    In house
     02
    (2R,3S,4S,5S)-5-羥基-2,3,4-三 (芐氧基)-5-[(芐氧基)甲基]-環己酮 (2R,3S,4S,5S)-5-Hydroxy-2,3,4-tris (phenylmethoxy)-5-[(phenylmethoxy)methyl]-cyclohexanone115250-38-9≥99%
    In house
     03
    四芐基伏格列波糖
    Tetra-Benzyl-Voglibose
    115250-39-0≥99%
    In house
     04
    鹽酸吉西他濱中間體Gemcitabine Hydrochloride Intermediate2-脫氧-2,2二氟-戊呋喃糖-1-酮- 3,5-二苯甲酸酯(T6) 2-Deoxy-2,2-difluoro-D-erythro-pentafuranous-1-ulose-3,5-dibenzoate122111-01-7≥99%
    In house
     05
    帕利哌酮及中間體
    Paliperidone & Intermediates
    帕利哌酮
    Paliperidone
    144598-75-4≥99%
    In house
     06
    帕利哌酮棕櫚酸酯
    Paliperidone Palmitate
    199739-10-1≥99%
    In house
     07
    3-(2-氯乙基)-6,7,8,9-四氫-9-羥基-2-甲基-4H-吡啶并[1,2-a]嘧啶-4-酮3-(2-Chloroethyl)-6,7,8,9-tetrahydro-9-hydroxy-2-methyl-4H-pyrido[1,2-a]pyrimidin-4-one130049-82-0≥99%
    In house
     08
    6-氟-3-哌啶-4-基-1,2-苯并異噁唑鹽酸鹽
    6-Fluoro-3-(4-piperidinyl)-1,2-
    benzisoxazole hydrochloride
    84163-13-3≥99%
    In house
     09
    鹽酸厄洛替尼中間體
    Erlotinib Hydrochloride
    Intermediates
    6,7-雙(甲氧基乙氧基)喹唑啉酮
    6,7-Bis-(2-methoxyethoxy)-4(3H)-quinazolinone
    179688-29-0≥99%
    In house
     10
    阿加曲班及中間體Argatroban &
    Intermediate
    阿加曲班
    Argatroban Hydrate
    74863-84-6≥99%
    In house
     11
    (2R,4R)-4-甲基-2-哌啶甲酸乙酯
    Ethyl (2R,4R)-4-methyl-2-piperidinecarboxylate
    74892-82-3≥99%
         In house
     12
    帕布昔利布及中間體Palbociclib & Intermediates帕布昔利布(帕博西尼)
    Palbociclib
    571190-30-2≥99%
    In house
     13
    4-(6-氨基吡啶-3-基)哌嗪-1-羧酸叔丁酯
    4-(6-Aminopyridin-3-yl)piperazine-1-carboxylic acid tert-butyl este
    571188-59-5≥99%
    In house
     14
    6-溴-2-氯-8-環戊基-5-甲基-吡啶并[2,3-D]嘧啶-7(8H)-酮6-bromo-2-chloro-8-cyclopentyl-5-Methylpyrido[2,3-d]pyriMidin-7(8H)-one1016636-76-2≥99%
    In house
     15
    奧格列汀Omarigliptin & IntermediatesN-[(2R,3S)-2-(2,5-二氟苯基)四氫-5-氧代-2H-吡喃-3-基]氨基甲酸叔丁酯N-[(2R,3S)-2-(2,5-Difluorophenyl)tetrahydro-5-oxo-2H-pyran-3-yl]carbamic acid 1,1-dimethylethyl ester951127-25-6≥99%
    In house
     16
    2-(甲基磺?;?-2,4,5,6-四氫吡咯并[3,4-c]吡唑苯磺酸鹽
    2,4,5,6-Tetrahydro-2-(methylsulfonyl)pyrrolo[3,4-c]pyrazole benzenesulfonate
    1280210-80-1≥99%
    In house
     17


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